CRYSTAL STRUCTURE OF JAK3 KINASE DOMAIN IN COMPLEX WITH A PYRROLOPYRIDAZINE INHIBITOR
收藏Protein Data Bank Japan2024-03-13 更新2026-03-21 收录
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https://pdbj.org/mine/summary/5vo6
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CRYSTAL STRUCTURE OF JAK3 KINASE DOMAIN IN COMPLEX WITH A PYRROLOPYRIDAZINE INHIBITOR Descriptor: 4-{[(1R,3S)-3-amino-2,2,3-trimethylcyclopentyl]amino}-6-phenylpyrrolo[1,2-b]pyridazine-3-carboxamide, Tyrosine-protein kinase JAK3 Authors: Sack, J.S. Deposit date: 2017-05-02 Release date: 2017-05-31 Last modified: 2024-03-13 Method: X-RAY DIFFRACTION (2.65 Å) Cite: Discovery of potent and efficacious pyrrolopyridazines as dual JAK1/3 inhibitors. Bioorg. Med. Chem. Lett., 27, 2017
创建时间:
2017-05-02



