Crystal structure of the first bromodomain (BD1) of human BRD2 bound to volasertib
收藏Protein Data Bank Japan2023-10-18 更新2026-03-21 收录
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Crystal structure of the first bromodomain (BD1) of human BRD2 bound to volasertib Descriptor: Bromodomain-containing protein 2, N-{trans-4-[4-(cyclopropylmethyl)piperazin-1-yl]cyclohexyl}-4-{[(7R)-7-ethyl-5-methyl-8-(1-methylethyl)-6-oxo-5,6,7,8-tetrahydropteridin-2-yl]amino}-3-methoxybenzamide Authors: Karim, M.R, Bikowitz, M, Chan, A, Schonbrunn, E. Deposit date: 2021-01-06 Release date: 2021-07-14 Last modified: 2023-10-18 Method: X-RAY DIFFRACTION (1.831 Å) Cite: Differential BET Bromodomain Inhibition by Dihydropteridinone and Pyrimidodiazepinone Kinase Inhibitors. J.Med.Chem., 64, 2021
创建时间：
2021-01-06
