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CRYSTAL STRUCTURE OF NAMPT IN COMPLEX WITH COMPOUND 9

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Protein Data Bank Japan2024-01-31 更新2026-03-28 收录
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https://pdbj.org/mine/summary/7ppg
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资源简介:
CRYSTAL STRUCTURE OF NAMPT IN COMPLEX WITH COMPOUND 9 Descriptor: 1,2-ETHANEDIOL, N-[4-[(4R)-1-cyclopentyl-4-methyl-6-oxidanylidene-4,5-dihydropyridazin-3-yl]phenyl]-1,3-dihydropyrrolo[3,4-c]pyridine-2-carboxamide, Nicotinamide phosphoribosyltransferase, ... Authors: Hillig, R.C. Deposit date: 2021-09-13 Release date: 2022-06-15 Last modified: 2024-01-31 Method: X-RAY DIFFRACTION (2.13 Å) Cite: A Novel NAMPT Inhibitor-Based Antibody-Drug Conjugate Payload Class for Cancer Therapy. Bioconjug.Chem., 33, 2022
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2021-09-13
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