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Crystal Structure Analysis of a 6-Amino Quinazolinedione Sulfonamide bound to human GluR2

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Protein Data Bank Japan2024-11-20 更新2026-03-21 收录
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Crystal Structure Analysis of a 6-Amino Quinazolinedione Sulfonamide bound to human GluR2 Descriptor: Glutamate receptor 2, N-methyl-1-{3-[(methylsulfonyl)amino]-2,4-dioxo-7-(trifluoromethyl)-1,2,3,4-tetrahydroquinazolin-6-yl}-1H-imidazole-4-carboxamide Authors: Kallen, J. Deposit date: 2011-10-21 Release date: 2012-01-11 Last modified: 2024-11-20 Method: X-RAY DIFFRACTION (1.9 Å) Cite: 6-Amino quinazolinedione sulfonamides as orally active competitive AMPA receptor antagonists. Bioorg.Med.Chem.Lett., 22, 2012
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2011-10-21
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