Structure of CHK1 10-pt. mutant complex with LRRK2 inhibitor 18
收藏Protein Data Bank Japan2023-10-18 更新2026-03-21 收录
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Structure of CHK1 10-pt. mutant complex with LRRK2 inhibitor 18 Descriptor: N-{5-[(3S)-3-(2-hydroxypropan-2-yl)pyrrolidin-1-yl]-2-(trifluoromethyl)pyridin-3-yl}-6-(1-methyl-1H-pyrazol-4-yl)pyridine-2-carboxamide, Serine/threonine-protein kinase Chk1 Authors: Palte, R. Deposit date: 2021-04-02 Release date: 2021-06-16 Last modified: 2023-10-18 Method: X-RAY DIFFRACTION (1.65 Å) Cite: Optimization of brain-penetrant picolinamide derived leucine-rich repeat kinase 2 (LRRK2) inhibitors. Rsc Med Chem, 12, 2021
创建时间:
2021-04-02



