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TBK1 in complex with Inhibitor compound 35

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Protein Data Bank Japan2024-01-24 更新2026-03-21 收录
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TBK1 in complex with Inhibitor compound 35 Descriptor: 3,3,3-tris(fluoranyl)-1-[4-[(1~{R})-1-[2-[[(2~{S})-5-(5-propan-2-yloxypyrimidin-4-yl)-2,3-dihydro-1~{H}-benzimidazol-2-yl]amino]pyridin-4-yl]ethyl]piperazin-1-yl]propan-1-one, Serine/threonine-protein kinase TBK1 Authors: Panne, D, Hillig, R.C, Rengachari, S. Deposit date: 2019-05-22 Release date: 2020-04-01 Last modified: 2024-01-24 Method: X-RAY DIFFRACTION (2.75 Å) Cite: Discovery of BAY-985, a Highly Selective TBK1/IKK epsilon Inhibitor. J.Med.Chem., 63, 2020

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2019-05-22
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