DCN1 bound to DI-1548
收藏Protein Data Bank Japan2024-10-16 更新2026-03-21 收录
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DCN1 bound to DI-1548 Descriptor: Lysozyme, DCN1-like protein 1 chimera, N-{(1S)-1-cyclohexyl-2-[(2-methylpropanoyl)amino]ethyl}-N~2~-propanoyl-3-[6-(propan-2-yl)-1,3-benzothiazol-2-yl]-L-alaninamide Authors: Stuckey, J.A. Deposit date: 2020-07-07 Release date: 2021-06-02 Last modified: 2024-10-16 Method: X-RAY DIFFRACTION (2.39 Å) Cite: Selective inhibition of cullin 3 neddylation through covalent targeting DCN1 protects mice from acetaminophen-induced liver toxicity. Nat Commun, 12, 2021
创建时间:
2020-07-07



