five

mPI3Kd in complex with compound 58

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Protein Data Bank Japan2024-05-01 更新2026-03-28 收录
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mPI3Kd in complex with compound 58 Descriptor: 2-[(1S)-1-cyclopropylethyl]-5-[4-methyl-2-[[6-(2-oxidanylidenepyrrolidin-1-yl)pyridin-2-yl]amino]-1,3-thiazol-5-yl]-7-methylsulfonyl-3H-isoindol-1-one, Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform, SODIUM ION Authors: Petersen, J. Deposit date: 2021-05-11 Release date: 2021-07-14 Last modified: 2024-05-01 Method: X-RAY DIFFRACTION (1.95 Å) Cite: Discovery of AZD8154, a Dual PI3K gamma delta Inhibitor for the Treatment of Asthma. J.Med.Chem., 64, 2021
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2021-05-11
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