Crystal Structure of EHMT2 bound to EZM8266
收藏Protein Data Bank Japan2025-07-23 更新2026-05-23 收录
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Crystal Structure of EHMT2 bound to EZM8266 Descriptor: (2R)-1-(azetidin-1-yl)-3-(2-methoxy-5-{[4-methyl-6-(methylamino)pyrimidin-2-yl]amino}phenoxy)propan-2-ol, Histone-lysine N-methyltransferase EHMT2, S-ADENOSYLMETHIONINE, ... Authors: Cocozaki, A, Farrow, N.A. Deposit date: 2024-01-30 Release date: 2024-12-11 Last modified: 2025-07-23 Method: X-RAY DIFFRACTION (2 Å) Cite: Combining EHMT and PARP Inhibition: A Strategy to Diminish Therapy-Resistant Ovarian Cancer Tumor Growth while Stimulating Immune Activation. Mol.Cancer Ther., 23, 2024
创建时间:
2024-01-30



