HUMAN JAK3 IN COMPLEX WITH LASW959 PROTEIN IN COMPLEX WITH LIGAND
收藏Protein Data Bank Japan2024-11-06 更新2026-03-21 收录
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HUMAN JAK3 IN COMPLEX WITH LASW959 PROTEIN IN COMPLEX WITH LIGAND Descriptor: 3-[7-(2-hydroxyethyl)-9-(oxan-4-yl)-8-oxidanylidene-purin-2-yl]imidazo[1,2-a]pyridine-6-carbonitrile, Tyrosine-protein kinase JAK3 Authors: Lozoya, E, Segarra, V, Bach, J, Jestel, A, Lammens, A, Blaesse, M. Deposit date: 2018-10-24 Release date: 2019-10-23 Last modified: 2024-11-06 Method: X-RAY DIFFRACTION (2.46 Å) Cite: Identification of 2-Imidazopyridine and 2-Aminopyridone Purinones as Potent Pan-Janus Kinase (JAK) Inhibitors for the Inhaled Treatment of Respiratory Diseases. J.Med.Chem., 62, 2019
创建时间:
2018-10-24



