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STRUCTURE OF MCL1 BOUND TO BRD inhibitor ligand 1 AT 1.7A

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Protein Data Bank Japan2023-12-27 更新2026-03-21 收录
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STRUCTURE OF MCL1 BOUND TO BRD inhibitor ligand 1 AT 1.7A Descriptor: 7-[2-(1H-imidazol-1-yl)-4-methylpyridin-3-yl]-3-[3-(naphthalen-1-yloxy)propyl]-1-[2-oxo-2-(piperazin-1-yl)ethyl]-1H-indole-2-carboxylic acid, Induced myeloid leukemia cell differentiation protein Mcl-1, PYROPHOSPHATE 2-, ... Authors: CLIFTON, M.C, EDWARDS, T.E. Deposit date: 2014-10-09 Release date: 2015-05-06 Last modified: 2023-12-27 Method: X-RAY DIFFRACTION (1.7 Å) Cite: A Maltose-Binding Protein Fusion Construct Yields a Robust Crystallography Platform for MCL1. Plos One, 10, 2015

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2014-10-09
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