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Crystal structure of NUDT1 (MTH1) with S-crizotinib

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Protein Data Bank Japan2023-12-20 更新2026-03-21 收录
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Crystal structure of NUDT1 (MTH1) with S-crizotinib Descriptor: 3-[(1S)-1-(2,6-DICHLORO-3-FLUOROPHENYL)ETHOXY]-5-(1-PIPERIDIN-4-YLPYRAZOL-4-YL)PYRIDIN-2-AMINE, 7,8-DIHYDRO-8-OXOGUANINE TRIPHOSPHATASE, CHLORIDE ION, ... Authors: Elkins, J.M, Salah, E, Huber, K, Superti-Furga, G, Abdul Azeez, K.R, Krojer, T, von Delft, F, Bountra, C, Edwards, A, Knapp, S. Deposit date: 2013-10-03 Release date: 2014-04-02 Last modified: 2023-12-20 Method: X-RAY DIFFRACTION (1.2 Å) Cite: Stereospecific Targeting of Mth1 by (S)-Crizotinib as an Anticancer Strategy. Nature, 508, 2014
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2013-10-03
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