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Crystal structure of JAK2 JH2-V617F in complex with Reversine

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Protein Data Bank Japan2024-10-16 更新2026-04-25 收录
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https://pdbj.org/mine/summary/8bak
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Crystal structure of JAK2 JH2-V617F in complex with Reversine Descriptor: GLYCEROL, N~6~-cyclohexyl-N~2~-(4-morpholin-4-ylphenyl)-9H-purine-2,6-diamine, Tyrosine-protein kinase JAK2 Authors: Haikarainen, T, Silvennoinen, O. Deposit date: 2022-10-11 Release date: 2023-02-01 Last modified: 2024-10-16 Method: X-RAY DIFFRACTION (1.65 Å) Cite: Identification of Novel Small Molecule Ligands for JAK2 Pseudokinase Domain. Pharmaceuticals, 16, 2023
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2022-10-11
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