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Discovery of Lysine-Targeted eIF4E Inhibitors through Covalent Docking

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Protein Data Bank Japan2024-10-16 更新2026-03-21 收录
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Discovery of Lysine-Targeted eIF4E Inhibitors through Covalent Docking Descriptor: 3-{(1-oxo-1,2-dihydroisoquinolin-7-yl)[(pyridin-4-yl)methyl]sulfamoyl}benzene-1-sulfonyl fluoride, Eukaryotic translation initiation factor 4E Authors: Wan, X.B, Shoichet, B.K, Taunton, J. Deposit date: 2019-08-13 Release date: 2019-10-23 Last modified: 2024-10-16 Method: X-RAY DIFFRACTION (1.79 Å) Cite: Discovery of Lysine-Targeted eIF4E Inhibitors through Covalent Docking. J.Am.Chem.Soc., 142, 2020

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2019-08-13
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