遇见数据集

STRUCTURE OF AURORA A IN COMPLEX WITH MLN8054

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Protein Data Bank Japan2023-12-20 更新2026-03-21 收录
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STRUCTURE OF AURORA A IN COMPLEX WITH MLN8054 Descriptor: 4-{[9-CHLORO-7-(2,6-DIFLUOROPHENYL)-5H-PYRIMIDO[5,4-D][2]BENZAZEPIN-2-YL]AMINO}BENZOIC ACID, SERINE/THREONINE-PROTEIN KINASE 6 Authors: Savory, W, Mueller, I, Mason, C.S, Lamers, M, Williams, D.H, Eyers, P.A. Deposit date: 2010-03-05 Release date: 2010-05-05 Last modified: 2023-12-20 Method: X-RAY DIFFRACTION (2.91 Å) Cite: Drug-Resistant Aurora a Mutants for Cellular Target Validation of the Small Molecule Kinase Inhibitors Mln8054 and Mln8237. Acs Chem.Biol., 5, 2010

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2010-03-05
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