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Crystal Structure of PDE10A with Novel Keto-Benzimidazole Inhibitor

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Protein Data Bank Japan2024-11-27 更新2026-03-21 收录
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Crystal Structure of PDE10A with Novel Keto-Benzimidazole Inhibitor Descriptor: 1H-benzimidazol-2-yl(4-{[3-(morpholin-4-yl)pyrazin-2-yl]oxy}phenyl)methanone, SULFATE ION, ZINC ION, ... Authors: Chmait, S, Jordan, S. Deposit date: 2013-09-24 Release date: 2013-10-23 Last modified: 2024-11-27 Method: X-RAY DIFFRACTION (2.496 Å) Cite: Design, Optimization, and Biological Evaluation of Novel Keto-Benzimidazoles as Potent and Selective Inhibitors of Phosphodiesterase 10A (PDE10A). J.Med.Chem., 56, 2013

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2013-09-24
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