Quadruple mutant plasmodium falciparum dihydrofolate reductase complexed with B10042
收藏Protein Data Bank Japan2023-11-22 更新2026-03-21 收录
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https://pdbj.org/mine/summary/6kp2
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Quadruple mutant plasmodium falciparum dihydrofolate reductase complexed with B10042 Descriptor: 5-(3-chlorophenyl)-6-(3-phenoxypropyl)pyrimidine-2,4-diamine, Bifunctional dihydrofolate reductase-thymidylate synthase, GLYCEROL, ... Authors: Vanichtanankul, J, Vitsupakorn, D. Deposit date: 2019-08-14 Release date: 2019-12-04 Last modified: 2023-11-22 Method: X-RAY DIFFRACTION (1.973 Å) Cite: 6-Hydrophobic aromatic substituent pyrimethamine analogues as potential antimalarials for pyrimethamine-resistant Plasmodium falciparum. Bioorg.Med.Chem., 27, 2019
创建时间:
2019-08-14



