Crystal structure of GSK3b in complex with N-(4-(5-(1,2,4-oxadiazol-3-yl)thiophen-2-yl)pyridin-2-yl)cyclopropanecarboxamide inhibitor (TW362)
收藏Protein Data Bank Japan2024-10-16 更新2026-04-19 收录
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Crystal structure of GSK3b in complex with N-(4-(5-(1,2,4-oxadiazol-3-yl)thiophen-2-yl)pyridin-2-yl)cyclopropanecarboxamide inhibitor (TW362) Descriptor: Glycogen synthase kinase-3 beta, N-[4-[5-(1,2,4-oxadiazol-3-yl)thiophen-2-yl]pyridin-2-yl]cyclopropanecarboxamide Authors: Slugocka, E.A, Grygier, P, Wichur, T, Czarna, A, Wieckowska, A. Deposit date: 2023-09-13 Release date: 2024-09-04 Last modified: 2024-10-16 Method: X-RAY DIFFRACTION (3.02 Å) Cite: Exploring Novel GSK-3 beta Inhibitors for Anti-Neuroinflammatory and Neuroprotective Effects: Synthesis, Crystallography, Computational Analysis, and Biological Evaluation. Acs Chem Neurosci, 15, 2024
创建时间:
2023-09-13



