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CRYSTAL STRUCTURE OF THE CATALYTIC DOMAIN OF HUMAN FIBROBLAST STROMELYSIN-1 INHIBITED WITH THIADIAZOLE INHIBITOR PNU-142372

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Protein Data Bank Japan2024-05-22 更新2026-03-21 收录
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CRYSTAL STRUCTURE OF THE CATALYTIC DOMAIN OF HUMAN FIBROBLAST STROMELYSIN-1 INHIBITED WITH THIADIAZOLE INHIBITOR PNU-142372 Descriptor: 2-[3-(5-MERCAPTO-[1,3,4]THIADIAZOL-2YL)-UREIDO]-N-METHYL-3-PENTAFLUOROPHENYL-PROPIONAMIDE, CALCIUM ION, STROMELYSIN-1, ... Authors: Finzel, B.C, Bryant Junior, G.L, Baldwin, E.T. Deposit date: 1998-06-09 Release date: 1998-12-23 Last modified: 2024-05-22 Method: X-RAY DIFFRACTION (1.8 Å) Cite: Structural characterizations of nonpeptidic thiadiazole inhibitors of matrix metalloproteinases reveal the basis for stromelysin selectivity. Protein Sci., 7, 1998
创建时间:
1998-06-09
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