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EGFR in complex with a dihydrodibenzodiazepinone allosteric inhibitor.

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Protein Data Bank Japan2023-10-11 更新2026-03-21 收录
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https://pdbj.org/mine/summary/6p8q
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EGFR in complex with a dihydrodibenzodiazepinone allosteric inhibitor. Descriptor: 1,2-ETHANEDIOL, 10-benzyl-2-fluoro-5,10-dihydro-11H-dibenzo[b,e][1,4]diazepin-11-one, ADENOSINE MONOPHOSPHATE, ... Authors: Yun, C.H, Heppner, D.E, Eck, M.J. Deposit date: 2019-06-07 Release date: 2019-12-18 Last modified: 2023-10-11 Method: X-RAY DIFFRACTION (1.9 Å) Cite: Discovery and Optimization of Dibenzodiazepinones as Allosteric Mutant-Selective EGFR Inhibitors. Acs Med.Chem.Lett., 10, 2019
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2019-06-07
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