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Low Micromolar Small Molecule Inhibitor of IL-2

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Protein Data Bank Japan2024-11-20 更新2026-03-21 收录
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Low Micromolar Small Molecule Inhibitor of IL-2 Descriptor: 2-CYCLOHEXYL-N-(2-{4-[5-(2,3-DICHLORO-PHENYL)-2H-PYRAZOL-3-YL]-PIPERIDIN-1-YL}-2-OXO-ETHYL)-2-GUANIDINO-ACETAMIDE, Interleukin-2, SULFATE ION Authors: Thanos, C.D, Randal, M, Wells, J.A. Deposit date: 2003-06-30 Release date: 2004-01-13 Last modified: 2024-11-20 Method: X-RAY DIFFRACTION (2.6 Å) Cite: Potent small-molecule binding to a dynamic hot spot on IL-2. J.Am.Chem.Soc., 125, 2003

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2003-06-30
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