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PvSub1 Catalytic Domain in Complex with Peptidomimetic Inhibitor (MAM-133)

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Protein Data Bank Japan2024-05-01 更新2026-04-19 收录
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PvSub1 Catalytic Domain in Complex with Peptidomimetic Inhibitor (MAM-133) Descriptor: 2-acetamido-2-deoxy-beta-D-glucopyranose, CALCIUM ION, Peptidomimetic Inhibitor (MAM-133), ... Authors: Batista, F.A, Martinez, M, Bouillon, A, Mechaly, A, Alzari, P.M, Haouz, A, Barale, J.C. Deposit date: 2023-09-15 Release date: 2024-03-20 Last modified: 2024-05-01 Method: X-RAY DIFFRACTION (1.767 Å) Cite: Insights from structure-activity relationships and the binding mode of peptidic alpha-ketoamide inhibitors of the malaria drug target subtilisin-like SUB1. Eur.J.Med.Chem., 269, 2024

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2023-09-15
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