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Crystal structure of the PDE4D catalytic domain in complex with GEBR-32a

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Protein Data Bank Japan2024-05-08 更新2026-03-21 收录
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Crystal structure of the PDE4D catalytic domain in complex with GEBR-32a Descriptor: (2~{R})-1-[3-[4-[bis(fluoranyl)methoxy]-3-cyclopentyloxy-phenyl]pyrazol-1-yl]-3-morpholin-4-yl-propan-2-ol, (2~{S})-1-[5-[4-[bis(fluoranyl)methoxy]-3-cyclopentyloxy-phenyl]pyrazol-1-yl]-3-morpholin-4-yl-propan-2-ol, 1,2-ETHANEDIOL, ... Authors: Prosdocimi, T, Donini, S, Parisini, E. Deposit date: 2017-12-22 Release date: 2018-05-16 Last modified: 2024-05-08 Method: X-RAY DIFFRACTION (1.45 Å) Cite: Molecular Bases of PDE4D Inhibition by Memory-Enhancing GEBR Library Compounds. Biochemistry, 57, 2018

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2017-12-22
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