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A crystal form of a human CDK2-CDK7 chimera

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Protein Data Bank Japan2024-08-21 更新2026-04-19 收录
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A crystal form of a human CDK2-CDK7 chimera Descriptor: (3R,4R)-4-[[[7-[(phenylmethyl)amino]-3-propan-2-yl-pyrazolo[1,5-a]pyrimidin-5-yl]amino]methyl]piperidin-3-ol, Cyclin-dependent kinase 2 Authors: Mukherjee, M, Cleasby, A. Deposit date: 2024-01-30 Release date: 2024-06-26 Last modified: 2024-08-21 Method: X-RAY DIFFRACTION (1.51 Å) Cite: Protein engineering enables a soakable crystal form of human CDK7 primed for high-throughput crystallography and structure-based drug design. Structure, 32, 2024

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2024-01-30
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