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Crystal structure of Retinoic Acid Receptor alpha (RXRA) in complexed with JP147

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Protein Data Bank Japan2024-02-21 更新2026-06-30 收录
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https://pdbj.org/mine/summary/8pp0
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Crystal structure of Retinoic Acid Receptor alpha (RXRA) in complexed with JP147 Descriptor: 3-[4-[2,3-dihydro-1H-inden-4-yl(methyl)amino]-6-(trifluoromethyl)pyrimidin-2-yl]oxypropanoic acid, Nuclear receptor coactivator 2, Retinoic acid receptor RXR-alpha Authors: Chaikuad, A, Pollinger, J, Merk, D, Knapp, S, Structural Genomics Consortium (SGC) Deposit date: 2023-07-05 Release date: 2024-02-07 Last modified: 2024-02-21 Method: X-RAY DIFFRACTION (1.9 Å) Cite: Structure-Guided Design of a Highly Potent Partial RXR Agonist with Superior Physicochemical Properties. J.Med.Chem., 67, 2024
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2023-07-05
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