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Crystal structure of Candida glabrata Bdf1 bromodomain 2 bound to I-BET151

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Protein Data Bank Japan2025-03-26 更新2026-04-19 收录
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Crystal structure of Candida glabrata Bdf1 bromodomain 2 bound to I-BET151 Descriptor: 7-(3,5-DIMETHYL-1,2-OXAZOL-4-YL)-8-METHOXY-1-[(1R)-1-(PYRIDIN-2-YL)ETHYL]-1H,2H,3H-IMIDAZO[4,5-C]QUINOLIN-2-ONE, Candida glabrata strain CBS138 chromosome C complete sequence, GLYCEROL, ... Authors: Petosa, C, Wei, K, McKenna, C.E, Govin, J. Deposit date: 2023-11-22 Release date: 2024-10-30 Last modified: 2025-03-26 Method: X-RAY DIFFRACTION (1.95 Å) Cite: Humanized Candida and NanoBiT Assays Expedite Discovery of Bdf1 Bromodomain Inhibitors With Antifungal Potential. Adv Sci, 12, 2025
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2023-11-22
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