Human Aurora A catalytic domain bound to FK1142
收藏Protein Data Bank Japan2024-01-10 更新2026-03-21 收录
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Human Aurora A catalytic domain bound to FK1142 Descriptor: (2Z,5Z)-2-[(4-ethylphenyl)imino]-3-methyl-5-[(2-{[4-(1H-tetrazol-5-yl)phenyl]amino}pyridin-4-yl)methylidene]-1,3-thiazolidin-4-one, (4S)-2-METHYL-2,4-PENTANEDIOL, Aurora kinase A Authors: Marcaida, M.J, Kilchmann, F, Schick, T, Reymond, J.L. Deposit date: 2015-05-15 Release date: 2016-07-20 Last modified: 2024-01-10 Method: X-RAY DIFFRACTION (2.9 Å) Cite: Discovery of a Selective Aurora A Kinase Inhibitor by Virtual Screening. J.Med.Chem., 59, 2016
创建时间:
2015-05-15



