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MBX3135 bound structure of bacterial efflux pump.

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Protein Data Bank Japan2024-05-08 更新2026-03-21 收录
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MBX3135 bound structure of bacterial efflux pump. Descriptor: DARPin, Multidrug efflux pump subunit AcrB,Multidrug efflux pump subunit AcrB, ~{N}-[4-[2-[[5-cyano-8-[(2~{S},6~{S})-2,6-dimethylmorpholin-4-yl]-3,3-dimethyl-1,4-dihydropyrano[3,4-c]pyridin-6-yl]sulfanyl]ethyl]phenyl]prop-2-enamide Authors: Sjuts, H, Ornik, A.R, Pos, K.M. Deposit date: 2015-11-09 Release date: 2016-04-06 Last modified: 2024-05-08 Method: X-RAY DIFFRACTION (2.3 Å) Cite: Molecular basis for inhibition of AcrB multidrug efflux pump by novel and powerful pyranopyridine derivatives. Proc.Natl.Acad.Sci.USA, 113, 2016

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2015-11-09
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