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Influenza polymerase basic protein 2 (PB2) bound to a small-molecule inhibitor

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Protein Data Bank Japan2023-09-20 更新2026-03-21 收录
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Influenza polymerase basic protein 2 (PB2) bound to a small-molecule inhibitor Descriptor: N~2~-[2-(5-chloro-1H-pyrrolo[2,3-b]pyridin-3-yl)-5-fluoropyrimidin-4-yl]-N,N-dimethyl-L-alaninamide, Polymerase basic protein 2 Authors: Jacobs, M.D. Deposit date: 2013-10-24 Release date: 2014-07-30 Last modified: 2023-09-20 Method: X-RAY DIFFRACTION (2.82 Å) Cite: Discovery of a Novel, First-in-Class, Orally Bioavailable Azaindole Inhibitor (VX-787) of Influenza PB2. J.Med.Chem., 57, 2014

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2013-10-24
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