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Crystal Structure Of AKR1B10 Complexed With NADP+ And Zopolrestat

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Protein Data Bank Japan2023-09-20 更新2026-03-21 收录
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Crystal Structure Of AKR1B10 Complexed With NADP+ And Zopolrestat Descriptor: 3,4-DIHYDRO-4-OXO-3-((5-TRIFLUOROMETHYL-2-BENZOTHIAZOLYL)METHYL)-1-PHTHALAZINE ACETIC ACID, Aldo-keto reductase family 1 member B10, NADP NICOTINAMIDE-ADENINE-DINUCLEOTIDE PHOSPHATE, ... Authors: Zhang, L, Zheng, X, Zhang, H, Zhao, Y, Chen, K, Zhai, J, Hu, X, Structural Genomics Consortium (SGC) Deposit date: 2013-03-06 Release date: 2013-10-23 Last modified: 2023-09-20 Method: X-RAY DIFFRACTION (2.2 Å) Cite: Inhibitor selectivity between aldo-keto reductase superfamily members AKR1B10 and AKR1B1: Role of Trp112 (Trp111). Febs Lett., 587, 2013
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2013-03-06
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