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Crystal structure of the human androgen receptor T877A mutant ligand-binding domain with cyproterone acetate

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Protein Data Bank Japan2023-08-30 更新2026-03-21 收录
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https://pdbj.org/mine/summary/2oz7
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Crystal structure of the human androgen receptor T877A mutant ligand-binding domain with cyproterone acetate Descriptor: Androgen receptor, CYPROTERONE ACETATE Authors: Bohl, C.E, Wu, Z, Miller, D.D, Bell, C.E, Dalton, J.T. Deposit date: 2007-02-25 Release date: 2007-03-27 Last modified: 2023-08-30 Method: X-RAY DIFFRACTION (1.8 Å) Cite: Crystal structure of the T877A human androgen receptor ligand-binding domain complexed to cyproterone acetate provides insight for ligand-induced conformational changes and structure-based drug design. J.Biol.Chem., 282, 2007
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2007-02-25
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