five

Structure of MELK in complex with inhibitors

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Protein Data Bank Japan2024-05-08 更新2026-03-21 收录
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Structure of MELK in complex with inhibitors Descriptor: 1-(4-{[3-(isoquinolin-7-yl)prop-2-yn-1-yl]oxy}-2-methoxybenzyl)piperazinediium, DIMETHYL SULFOXIDE, MATERNAL EMBRYONIC LEUCINE ZIPPER KINASE Authors: Johnson, C.N, Berdini, V, Beke, L, Bonnet, P, Brehmer, D, Coyle, J.E, Day, P.J, Frederickson, M, Freyne, E.J.E, Gilissen, R.A.H.J, Hamlett, C.C.F, Howard, S, Meerpoel, L, McMenamin, R, Patel, S, Rees, D.C, Sharff, A, Sommen, F, Wu, T, Linders, J.T.M. Deposit date: 2014-05-21 Release date: 2014-10-22 Last modified: 2024-05-08 Method: X-RAY DIFFRACTION (1.98 Å) Cite: Structure-Based Design of Type II Inhibitors Applied to Maternal Embryonic Leucine Zipper Kinase. Acs Med.Chem.Lett., 6, 2015
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2014-05-21
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