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Crystal structure of HPK1 in complex an inhibitor G1858

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Protein Data Bank Japan2024-03-13 更新2026-03-21 收录
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Crystal structure of HPK1 in complex an inhibitor G1858 Descriptor: Mitogen-activated protein kinase kinase kinase kinase 1, N-{2-(3,3-difluoropyrrolidin-1-yl)-6-[(3R)-pyrrolidin-3-yl]pyrimidin-4-yl}-1-(propan-2-yl)-1H-pyrazolo[4,3-c]pyridin-6-amine Authors: Wu, P, Lehoux, I, Mortara, K, Franke, Y, Chan, B.K, Wang, W. Deposit date: 2018-03-15 Release date: 2018-12-19 Last modified: 2024-03-13 Method: X-RAY DIFFRACTION (2.246 Å) Cite: Hematopoietic Progenitor Kinase-1 Structure in a Domain-Swapped Dimer. Structure, 27, 2019

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2018-03-15
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