Crystal Structure of Nur77 LBD in complex with N-(2'-(4-hydroxypiperidin-1-yl)-[4,4'-bipyridin]-2-yl)cinnamamide
收藏Protein Data Bank Japan2025-01-29 更新2026-06-30 收录
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Crystal Structure of Nur77 LBD in complex with N-(2'-(4-hydroxypiperidin-1-yl)-[4,4'-bipyridin]-2-yl)cinnamamide Descriptor: (~{E})-~{N}-[4-[2-(4-oxidanylpiperidin-1-yl)pyridin-4-yl]pyridin-2-yl]-3-phenyl-prop-2-enamide, Nuclear receptor subfamily 4immunitygroup A member 1 Authors: Hong, W.B, Lin, T.W. Deposit date: 2024-02-04 Release date: 2024-07-24 Last modified: 2025-01-29 Method: X-RAY DIFFRACTION (2.683 Å) Cite: Discovery of a novel exceptionally potent and orally active Nur77 ligand NB1 with a distinct binding mode for cancer therapy. Acta Pharm Sin B, 14, 2024
创建时间:
2024-02-04



