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SYK catalytic domain complexed with naphthyridine inhibitor

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Protein Data Bank Japan2024-03-06 更新2026-03-21 收录
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SYK catalytic domain complexed with naphthyridine inhibitor Descriptor: CHLORIDE ION, GLYCEROL, N-{7-[4-(dimethylamino)phenyl]-1,6-naphthyridin-5-yl}propane-1,3-diamine, ... Authors: Thoma, G, Veenstra, S, Strang, R, Blanz, J, Vangrevelinghe, E, Berghausen, J, Lee, C.C, Zerwes, H.-G. Deposit date: 2015-07-29 Release date: 2015-09-16 Last modified: 2024-03-06 Method: X-RAY DIFFRACTION (1.7 Å) Cite: Orally bioavailable Syk inhibitors with activity in a rat PK/PD model. Bioorg.Med.Chem.Lett., 25, 2015

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2015-07-29
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