遇见数据集

p53-Y220C Core Domain Covalently Bound to 5-Chloro-6-methylpyrazine-2-carbonitrile Soaked at 5 mM

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Protein Data Bank Japan2025-07-16 更新2026-08-24 收录
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p53-Y220C Core Domain Covalently Bound to 5-Chloro-6-methylpyrazine-2-carbonitrile Soaked at 5 mM Descriptor: 1,2-ETHANEDIOL, 4-(2-HYDROXYETHYL)-1-PIPERAZINE ETHANESULFONIC ACID, 5-chloranyl-6-methyl-pyrazine-2-carbonitrile, ... Authors: Stahlecker, J, Klett, T, Stehle, T, Boeckler, F.M. Deposit date: 2024-07-19 Release date: 2025-06-11 Last modified: 2025-07-16 Method: X-RAY DIFFRACTION (1.56 Å) Cite: S N Ar Reactive Pyrazine Derivatives as p53-Y220C Cleft Binders with Diverse Binding Modes. Drug Des Devel Ther, 19, 2025

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2024-07-19
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