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Crystal structure of M. tuberculosis DprE1 in complex with the non-covalent inhibitor QN129

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Protein Data Bank Japan2023-12-27 更新2026-03-21 收录
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Crystal structure of M. tuberculosis DprE1 in complex with the non-covalent inhibitor QN129 Descriptor: (2R)-2-{[(2R)-2-{[(2R)-2-hydroxypropyl]oxy}propyl]oxy}propan-1-ol, 3-[(4-cyanobenzyl)amino]-6-(trifluoromethyl)quinoxaline-2-carboxylic acid, FLAVIN-ADENINE DINUCLEOTIDE, ... Authors: Neres, J, Pojer, F, Cole, S.T. Deposit date: 2014-04-01 Release date: 2014-12-10 Last modified: 2023-12-27 Method: X-RAY DIFFRACTION (2.55 Å) Cite: 2-Carboxyquinoxalines Kill Mycobacterium tuberculosis through Noncovalent Inhibition of DprE1. Acs Chem.Biol., 10, 2015
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2014-04-01
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