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fragment-linked stabilizer for ERa - 14-3-3 interaction (AZ210)

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Protein Data Bank Japan2024-10-23 更新2026-05-23 收录
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fragment-linked stabilizer for ERa - 14-3-3 interaction (AZ210) Descriptor: 14-3-3 protein sigma, 4-[(2~{S})-3-azanyl-2-methyl-propyl]-7-methoxy-1-benzothiophene-2-carboximidamide, ERalpha peptide, ... Authors: Visser, E.J, Sijbesma, E, Ottmann, C. Deposit date: 2022-12-14 Release date: 2023-08-02 Last modified: 2024-10-23 Method: X-RAY DIFFRACTION (1.4 Å) Cite: From Tethered to Freestanding Stabilizers of 14-3-3 Protein-Protein Interactions through Fragment Linking. Angew.Chem.Int.Ed.Engl., 62, 2023

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2022-12-14
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