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Crystal structure of JAK2 JH2-V617F in complex with JNJ-7706621

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Protein Data Bank Japan2024-10-16 更新2026-05-23 收录
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Crystal structure of JAK2 JH2-V617F in complex with JNJ-7706621 Descriptor: 4-({5-amino-1-[(2,6-difluorophenyl)carbonyl]-1H-1,2,4-triazol-3-yl}amino)benzenesulfonamide, GLYCEROL, Tyrosine-protein kinase JAK2 Authors: Haikarainen, T, Silvennoinen, O. Deposit date: 2022-10-05 Release date: 2023-02-01 Last modified: 2024-10-16 Method: X-RAY DIFFRACTION (1.6 Å) Cite: Identification of Novel Small Molecule Ligands for JAK2 Pseudokinase Domain. Pharmaceuticals, 16, 2023

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2022-10-05
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