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PARP15 catalytic domain in complex with OUL228

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Protein Data Bank Japan2024-01-31 更新2026-03-28 收录
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PARP15 catalytic domain in complex with OUL228 Descriptor: 8-ethoxy-4~{H}-thieno[2,3-c]isoquinolin-5-one, DIMETHYL SULFOXIDE, Protein mono-ADP-ribosyltransferase PARP15 Authors: Maksimainen, M.M, Lehtio, L. Deposit date: 2021-06-14 Release date: 2021-12-08 Last modified: 2024-01-31 Method: X-RAY DIFFRACTION (1.95 Å) Cite: Analogs of TIQ-A as inhibitors of human mono-ADP-ribosylating PARPs. Bioorg.Med.Chem., 52, 2021

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2021-06-14
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