Crystal structure of SETDB1 Tudor domain in complex with MR46747
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Crystal structure of SETDB1 Tudor domain in complex with MR46747 Descriptor: (3S)-N-(4-chloro-3-{[2-(diethylamino)ethyl]carbamoyl}phenyl)-3-(diethylamino)pyrrolidine-1-carboxamide, 1,2-ETHANEDIOL, Histone-lysine N-methyltransferase SETDB1, ... Authors: Shrestha, S, Beldar, S, Dong, A, Ackloo, S, Brown, P.J, Arrowsmith, C.H, Edwards, A.M, Halabelian, L, Structural Genomics Consortium (SGC) Deposit date: 2023-11-07 Release date: 2023-11-22 Last modified: 2025-06-04 Method: X-RAY DIFFRACTION (1.77 Å) Cite: A Target Class Ligandability Evaluation of WD40 Repeat-Containing Proteins. J.Med.Chem., 68, 2025
创建时间:
2023-11-07



