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Structure of h-CHK1 complexed with A767085

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Protein Data Bank Japan2024-03-13 更新2026-03-21 收录
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Structure of h-CHK1 complexed with A767085 Descriptor: 3-(4'-HYDROXYBIPHENYL-4-YL)-N-(4-HYDROXYCYCLOHEXYL)-1,4-DIHYDROINDENO[1,2-C]PYRAZOLE-6-CARBOXAMIDE, Serine/threonine-protein kinase Chk1 Authors: Park, C. Deposit date: 2007-01-26 Release date: 2008-01-29 Last modified: 2024-03-13 Method: X-RAY DIFFRACTION (2.5 Å) Cite: Discovery of 1,4-dihydroindeno[1,2-c]pyrazoles as a novel class of potent and selective checkpoint kinase 1 inhibitors. Bioorg.Med.Chem., 15, 2007
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2007-01-26
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