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1.70 A resolution structure of SARS-CoV-2 3CL protease in complex with inhibitor 7j

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Protein Data Bank Japan2024-11-06 更新2026-03-21 收录
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1.70 A resolution structure of SARS-CoV-2 3CL protease in complex with inhibitor 7j Descriptor: (1S,2S)-2-[(N-{[(4,4-difluorocyclohexyl)methoxy]carbonyl}-L-leucyl)amino]-1-hydroxy-3-[(3S)-2-oxopyrrolidin-3-yl]propane-1-sulfonic acid, 3C-like proteinase, TETRAETHYLENE GLYCOL Authors: Lovell, S, Kashipathy, M.M, Battaile, K.P, Rathnayake, A.D, Zheng, J, Kim, Y, Nguyen, H.N, Chang, K.O, Groutas, W.C. Deposit date: 2020-06-30 Release date: 2020-07-08 Last modified: 2024-11-06 Method: X-RAY DIFFRACTION (1.7 Å) Cite: 3C-like protease inhibitors block coronavirus replication in vitro and improve survival in MERS-CoV-infected mice. Sci Transl Med, 12, 2020
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2020-06-30
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