five

ERK5 in complex with small molecule

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Protein Data Bank Japan2024-05-08 更新2026-03-21 收录
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ERK5 in complex with small molecule Descriptor: 4-({5-fluoro-4-[2-methyl-1-(propan-2-yl)-1H-imidazol-5-yl]pyrimidin-2-yl}amino)-N-[2-(piperidin-1-yl)ethyl]benzamide, GLYCEROL, Mitogen-activated protein kinase 7 Authors: Chen, H, Tucker, J, Wang, X, Gavine, P.R, Philips, C, Augustin, M.A, Schreiner, P, Steinbacher, S, Preston, M, Ogg, D. Deposit date: 2015-06-11 Release date: 2016-05-04 Last modified: 2024-05-08 Method: X-RAY DIFFRACTION (1.65 Å) Cite: Discovery of a novel allosteric inhibitor-binding site in ERK5: comparison with the canonical kinase hinge ATP-binding site. Acta Crystallogr D Struct Biol, 72, 2016
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2015-06-11
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