Human Brd2(BD2) mutant in complex with ET
收藏Protein Data Bank Japan2024-01-17 更新2026-03-21 收录
下载链接:
https://pdbj.org/mine/summary/5o3a
下载链接
链接失效反馈官方服务:
资源简介:
Human Brd2(BD2) mutant in complex with ET Descriptor: Bromodomain-containing protein 2, methyl (2R)-2-[(4S)-6-(4-chlorophenyl)-8-methoxy-1-methyl-4H-[1,2,4]triazolo[4,3-a][1,4]benzodiazepin-4-yl]butanoate Authors: Chan, K.-H, Runcie, A.C, Ciulli, A. Deposit date: 2017-05-23 Release date: 2018-02-14 Last modified: 2024-01-17 Method: X-RAY DIFFRACTION (2.4 Å) Cite: Optimization of a "bump-and-hole" approach to allele-selective BET bromodomain inhibition. Chem Sci, 9, 2018
创建时间:
2017-05-23



