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Co-crystal Structure of Toxoplasma gondii Prolyl tRNA Synthetase (TgPRS) in complex with L97 and L-pro

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Protein Data Bank Japan2023-11-29 更新2026-03-21 收录
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Co-crystal Structure of Toxoplasma gondii Prolyl tRNA Synthetase (TgPRS) in complex with L97 and L-pro Descriptor: 4-[(3S)-3-cyclopropyl-3-(hydroxymethyl)-2-oxidanylidene-pyrrolidin-1-yl]-N-[[3-fluoranyl-5-(1-methylpyrazol-4-yl)phenyl]methyl]-6-methyl-pyridine-2-carboxamide, PROLINE, Prolyl-tRNA synthetase (ProRS) Authors: Mishra, S, Malhotra, N, Yogavel, M, Sharma, A. Deposit date: 2021-07-06 Release date: 2022-09-28 Last modified: 2023-11-29 Method: X-RAY DIFFRACTION (2.42 Å) Cite: Targeting prolyl-tRNA synthetase via a series of ATP-mimetics to accelerate drug discovery against toxoplasmosis. Plos Pathog., 19, 2023
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2021-07-06
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