Crystal structure of the bromodomain of human CREBBP bound to the benzodiazepinone G02778174
收藏Protein Data Bank Japan2023-09-27 更新2026-03-21 收录
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Crystal structure of the bromodomain of human CREBBP bound to the benzodiazepinone G02778174 Descriptor: (4R)-N-benzyl-4-methyl-2-oxo-2,3,4,5-tetrahydro-1H-1,5-benzodiazepine-6-carboxamide, 1,2-ETHANEDIOL, CREB-binding protein, ... Authors: Jayaram, H, Poy, F, Setser, J.W, Bellon, S.F. Deposit date: 2016-02-18 Release date: 2016-04-20 Last modified: 2023-09-27 Method: X-RAY DIFFRACTION (1.05 Å) Cite: Fragment-Based Discovery of a Selective and Cell-Active Benzodiazepinone CBP/EP300 Bromodomain Inhibitor (CPI-637). Acs Med.Chem.Lett., 7, 2016
创建时间：
2016-02-18
