five

Crystal structure of Rnase L in complex with Sunitinib

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Protein Data Bank Japan2023-11-29 更新2026-03-21 收录
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Crystal structure of Rnase L in complex with Sunitinib Descriptor: 5'-O-MONOPHOSPHORYLADENYLYL(2'->5')ADENYLYL(2'->5')ADENOSINE, N-[2-(diethylamino)ethyl]-5-[(Z)-(5-fluoro-2-oxo-1,2-dihydro-3H-indol-3-ylidene)methyl]-2,4-dimethyl-1H-pyrrole-3-carbo xamide, PHOSPHATE ION, ... Authors: Tang, J, Huang, H. Deposit date: 2020-02-24 Release date: 2020-09-02 Last modified: 2023-11-29 Method: X-RAY DIFFRACTION (2.46 Å) Cite: Sunitinib inhibits RNase L by destabilizing its active dimer conformation. Biochem.J., 477, 2020
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2020-02-24
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