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Crystal structure of KPC-2 carbapenemase in complex with a phenyl boronic inhibitor.

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Protein Data Bank Japan2024-10-16 更新2026-03-21 收录
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Crystal structure of KPC-2 carbapenemase in complex with a phenyl boronic inhibitor. Descriptor: (~{E})-3-[2-(dihydroxyboranyl)phenyl]prop-2-enoic acid, Carbapenem-hydrolyzing beta-lactamase KPC Authors: Vicario, M, Celenza, G, Bellio, P, Perilli, M.G, Tondi, D, Cendron, L. Deposit date: 2016-11-21 Release date: 2018-03-14 Last modified: 2024-10-16 Method: X-RAY DIFFRACTION (1.5 Å) Cite: Phenylboronic Acid Derivatives as Validated Leads Active in Clinical Strains Overexpressing KPC-2: A Step against Bacterial Resistance. Chemmedchem, 13, 2018
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2016-11-21
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