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Crystal structure of pyruvate dehydrogenase kinase isoform 2 in complex with inhibitor PS2

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Protein Data Bank Japan2024-02-28 更新2026-03-21 收录
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Crystal structure of pyruvate dehydrogenase kinase isoform 2 in complex with inhibitor PS2 Descriptor: 4-(isoindolin-2-ylsulfonyl)benzene-1,3-diol, L(+)-TARTARIC ACID, [Pyruvate dehydrogenase [lipoamide]] kinase isozyme 2, ... Authors: Gui, W.J, Tso, S.C, Chuang, J.L, Wu, C.Y, Qi, X, Tambar, U.K, Wynn, R.M, Chuang, D.T. Deposit date: 2013-09-12 Release date: 2014-01-01 Last modified: 2024-02-28 Method: X-RAY DIFFRACTION (1.699 Å) Cite: Structure-guided Development of Specific Pyruvate Dehydrogenase Kinase Inhibitors Targeting the ATP-binding Pocket. J.Biol.Chem., 289, 2014
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2013-09-12
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